[PDF] academia.edu

[PDF][PDF] Optimal agonist/antagonist combinations maintain receptor response by preventing rapid b1-adrenergic receptor desensitization

R Lanzara - Int. J. Pharm, 2005 - academia.edu
… calculated to prevent receptor desensitization, which has … or as part of an agonist'antagonist
combination. The Iso and Dob … earliest events of receptor desensitization can be modeled …
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[HTML] bio-balance.com

[HTML][HTML] Preventing Rapid Receptor Desensitization at the β1-Adrenergic Receptor with Agonist/Antagonist Combinations

R Lanzara - CPS: medichem, 2003 - bio-balance.com
… agonist/antagonist combination solution to prevent desensitization. Both the Iso/Met and
Dob/Met agonist/antagonist combination … the earliest events of receptor desensitization can be …
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[PDF] bio-balance.com

Preventing Rapid Receptor Desensitization at the Β-Adrenergic Receptor with Agonist/Antagonist Combinations

R Lanzara - Science Direct Working Paper, 2003 - papers.ssrn.com
… agonist/antagonist combination solution to prevent desensitization. Both the Iso/Met and
Dob/Met agonist/antagonist combination … the earliest events of receptor desensitization can be …
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[PDF] bio-balance.com

[PDF][PDF] Preventing Rapid Receptor Desensitization at the>-Adrenergic Receptor with Agonist/Antagonist Combinations

R Lanzara - bio-balance.com
… agonist/antagonist combination solution to prevent desensitization. Both the Iso/Met and
Dob/Met agonist/antagonist combination … the earliest events of receptor desensitization can be …
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Partial dopamine agonists and dopaminergic stabilizers, in the treatment of psychosis

CA Tamminga, A Carlsson - Current Drug Targets-CNS & …, 2002 - ingentaconnect.com
… Moreover, the proportions of an agonist/antagonist combination can be varied to achieve an
… of these activities (presumably due to receptor desensitization) when administered over the …
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[HTML] karger.com

[HTML][HTML] The two formyl peptide receptors differently regulate GPR84-mediated neutrophil NADPH oxidase activity

J Mårtensson, M Sundqvist, A Manandhar… - Journal of Innate …, 2021 - karger.com
… for each agonist/antagonist combination is shown. c Naïve … experiments for each
agonist/antagonist combination is shown… terminated through homologous receptor desensitization …
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[PDF] archive.org

The Two Formyl Peptide Receptors Differently Regulate GPR84-Mediated Neutrophil NADPH Oxidase Activity

JMMSA Manandharb, LLL Zhangc, TUX Xiec… - 2021 - karger.com
… for each agonist/antagonist combination is shown. c Naïve … experiments for each
agonist/antagonist combination is shown… terminated through homologous receptor desensitization …
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[PDF] researchgate.net

Partial agonism of dopamine, serotonin and opiate receptors for psychiatry

F Yocca, CA Altar - Drug Discovery Today: Therapeutic Strategies, 2006 - Elsevier
… It is frequently administered with naloxone as an opioid partial agonist–antagonist combination
… , reducing the potential for receptor desensitization. When excessive neurotransmission …
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[HTML] nih.gov

[HTML][HTML] 5-HT2A receptor activation normalizes exaggerated fear behavior in p-chlorophenylalanine (PCPA)-treated rats

CR Hughes, L Tran, NB Keele - Journal of behavioral and brain …, 2012 - ncbi.nlm.nih.gov
… Factor 2 (4 drug conditions, within groups) was the agonist/antagonist combination given
on … inhibition of fear may also involve receptor desensitization. While the amygdala seems a …
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[HTML][HTML] Gonadotropin-releasing hormone receptors in prostate cancer: molecular aspects and biological functions

F Fontana, M Marzagalli, M Montagnani Marelli… - International journal of …, 2020 - mdpi.com
… Interestingly, according to Uemura and coworkers, GnRH agonist/antagonist combination
treatments represent the mainstay therapeutic approach in CRPC patients in Japan [185]. …
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